Plant Growth Regulator Daminozide Is a Selective Inhibitor of Human KDM2/7 Histone Demethylases

Rose NR., Woon ECY., Tumber A., Walport LJ., Chowdhury R., Li XS., King ONF., Lejeune C., Ng SS., Krojer T., Chan MC., Rydzik AM., Hopkinson RJ., Che KH., Daniel M., Strain-Damerell C., Gileadi C., Kochan G., Leung IKH., Dunford J., Yeoh KK., Ratcliffe PJ., Burgess-Brown N., von Delft F., Muller S., Marsden B., Brennan PE., McDonough MA., Oppermann U., Klose RJ., Schofield CJ., Kawamura A.

DOI

10.1021/jm300677j

Type

Journal article

Journal

Journal of Medicinal Chemistry

Publisher

American Chemical Society (ACS)

Publication Date

26/07/2012

Volume

55

Pages

6639 - 6643

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