Linking of 2-Oxoglutarate and Substrate Binding Sites Enables Potent and Highly Selective Inhibition of JmjC Histone Demethylases

Woon ECY., Tumber A., Kawamura A., Hillringhaus L., Ge W., Rose NR., Ma JHY., Chan MC., Walport LJ., Che KH., Ng SS., Marsden BD., Oppermann U., McDonough MA., Schofield CJ.

DOI

10.1002/anie.201107833

Type

Journal article

Journal

Angewandte Chemie International Edition

Publisher

Wiley

Publication Date

13/02/2012

Volume

51

Pages

1631 - 1634

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